Bifeprunox 602S R S)-AHPC-Me-CO-CH2-PEG3-NH2 15(19)-tetraen-3-yl 1-methyl (3R)-3-hydroxy-3-(3-hydroxy-3-methylbutyl)butanedioate

15(19)-tetraen-3-yl 1-methyl (3R)-3-hydroxy-3-(3-hydroxy-3-methylbutyl)butanedioate

Vorapaxar (SCH 530348) inhibits thrombininduced calcium transient in human coronary artery smooth muscle cells (HCASMC) with a Ki of 1

it is observed that GSK4716 induces the expression of the mRNAs encoding peroxisome proliferator-activated receptor-γcoactivator 1α (PGC-1α) and PGC-1β (key regulator of many metabolic genes) identified as direct coactivators for the ERR family

there is a growth arrest and inhibition of DNA synthesis

CAS Number: 103-81-1

Bifeprunox 602S R S)-AHPC-Me-CO-CH2-PEG3-NH2 15(19)-tetraen-3-yl 1-methyl (3R)-3-hydroxy-3-(3-hydroxy-3-methylbutyl)butanedioateBifeprunox is a potent dopamine D2 like and 5 HT1A receptor partial agonist with pKis of 7. 19 and 8. 83 for cortex 5 HT1A and striatum D2, and a pEC50 of 6. 37 for hippocampus 5 HT1A, respectively. Bifeprunox is an antipsychotic for the research of schizophrenia. Product information CAS Number: 350992 10 8 Molecular Weight: 385. 46 Formula: C24H23N3O2 Chemical Name: 7 [4 ({[1,1' biphenyl] 3 yl}methyl)piperazin 1 yl] 2,3 dihydro 1,3 benzoxazol 2 one