In one of the experiments
EW-7197 Hydrochloride abolishes the TGFβ1-induced effects on genes related to epithelial-to-mesenchymal transition (EMT)
Entecavir-triphosphate is a highly potent inhibitor of wild-type HBV Pol and is 100- to 300-fold more potent than lamivudine-triphosphate against 3TC-resistant HBV Pol
IQ-1S free acid has binding affinity (Kd values) in the nanomolar range for all three JNKs with Kds of 100 nM
Chemical Name: propyl 2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]-[1
I-BET282 ts-2 In one of the experimentsI BET282 is a pan inhibitor of all eight BET bromodomains, and selectivity over other representative bromodomain containing proteins. I BET282 shows pIC50s ranging 6. 4 7. 7 for BRD2 (BD1 BD2), BRD2 (BD1 BD), BRD3 (BD1 BD), and BRD4 (BD1 BD). Product information CAS Number: 1422554 34 4 Molecular Weight: 450. 53 Formula: C25H30N4O4 Chemical Name: 4 {8 methoxy 1 [(2R) 1 methoxypropan 2 yl] 2 (oxan 4 yl) 1H imidazo[4,5 c]quinolin 7 yl} 3,5 dimethyl 1,2